Dragon Pharma
Dragon Pharma
Trestolone 100 mg
Product Information Compound Details
Active Substance Trestolone Enanthate Long-acting 19-nor testosterone derivative (MENT)
100 mg/mLStrength 100 mg/mL
Package 10 mL Vial 1,000 mg total labeled content
Form Oil-Based Injectable
Carrier MCT Oil
Drug Class Anabolic Androgenic Steroid (19-nor)
Manufacturer Dragon Pharma
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Product Overview
Trestolone 100 mg by Dragon Pharma
Trestolone 100 mg is an oil-based Trestolone Enanthate injectable manufactured by Dragon Pharma and dosed at 100 mg/mL in a 10 mL vial.
Trestolone Enanthate Injectable
Trestolone 100 mg contains trestolone enanthate, the long-acting enanthate ester of trestolone (7α-methyl-19-nortestosterone, or MENT). Trestolone is a synthetic anabolic-androgenic steroid derived from nandrolone, developed by the Population Council as a potential male hormonal contraceptive. The enanthate ester is a long-chain fatty acid attached to the 17-beta hydroxyl group that slows release from the injection site, extending the compound's active life to approximately 8 days according to pharmacological data.
Trestolone was investigated extensively as a candidate for hormonal male contraception and androgen replacement therapy, with clinical studies demonstrating that regular administration induces a state of temporary infertility by suppressing luteinizing hormone and follicle-stimulating hormone. Despite promising preclinical and early clinical data, trestolone and its esters have not received regulatory approval for medical use owing to concerns over side effects, including potential impacts on prostate health and lipid profiles. In non-medical bodybuilding contexts, Trestolone 100 mg is commonly referenced for its exceptional anabolic potency and rapid body recomposition effects.
Trestolone is notable for its resistance to 5α-reductase, meaning it does not convert to a DHT-like metabolite and is considered less prone to causing prostate enlargement compared to testosterone. However, it is a potent aromatase substrate that converts to 7α-methylestradiol (mestranol), a highly potent estrogen with effects that may bypass standard aromatase inhibitors. This estrogenic activity is frequently cited as the primary consideration when using the compound in non-medical contexts. Trestolone enanthate has an elimination half-life of about 8 days, allowing for less frequent injections compared to the acetate ester.
Key Benefits of Trestolone 100 mg
- Long-acting enanthate ester for less frequent injections
- Extremely potent anabolic activity with high anabolic-to-androgenic ratio
- Does not convert to DHT due to 5α-reductase resistance
- Commonly referenced for rapid muscle and strength gains
- MCT oil carrier for smooth injection
Carrier Oil
MCT Oil Formulation
Trestolone 100 mg uses MCT oil as its carrier, providing an oil base for the trestolone enanthate formulation. The 100 mg/mL concentration is a standard strength for this compound, allowing for practical injection volumes at commonly referenced doses.
Product Profile
Trestolone Enanthate Profile
Trestolone enanthate is a long-acting 19-nor anabolic steroid with exceptional anabolic potency and unique pharmacological characteristics. Its resistance to 5α-reductase and potent aromatization distinguish it from other injectable AAS compounds.
Potent 19-nor Anabolic Steroid (MENT)
Trestolone is structurally derived from nandrolone with a methyl group at the C7α position, which confers resistance to 5α-reductase and increases receptor affinity. Preclinical studies have demonstrated that trestolone exhibits approximately ten times the anabolic potency of testosterone, making it one of the most powerful AAS investigated. Its anabolic-to-androgenic ratio is reported to be approximately 600:200 when compared to testosterone's baseline of 100:100.
The compound binds to the androgen receptor with high affinity and, unlike testosterone, has low affinity for sex hormone-binding globulin (SHBG), which means a greater percentage of the administered dose remains available for receptor interaction. This contributes to its potency at relatively low doses compared to other injectable AAS. Trestolone enanthate serves as a depot formulation that prolongs the release and action of the active compound, with an elimination half-life of about 8 days.
Trestolone was studied as a male contraceptive, with clinical research demonstrating that sufficient quantities induce temporary infertility by suppressing gonadotropin release. The enanthate ester was specifically developed to provide a longer-acting injectable formulation for these applications.
Release Profile
Extended Trestolone Release
The enanthate ester of Trestolone 100 mg produces a longer duration of action than the acetate ester, with an elimination half-life of approximately 8 days. In non-medical contexts, this allows for injections once or twice per week, though some users prefer more frequent administration for stable blood levels. The slower release means that blood levels build gradually over several weeks, and side effects, if they occur, may persist longer after discontinuation compared to the acetate ester. Forum discussions reference that trestolone enanthate takes approximately 2 weeks to begin noticeable effects, with full saturation occurring over 4-5 weeks.
Trestolone 100 mg vs Other Dragon Pharma Preparations
Dragon Pharma offers a shorter-acting version of this compound, Ment 50, which contains trestolone acetate at 50 mg/mL and provides a more rapid onset and clearance. The enanthate ester in Trestolone 100 mg is better suited for users who prefer less frequent injections and more stable blood levels. For those seeking a traditional 19-nor compound with a different side effect profile, Deca 300 (nandrolone decanoate) is a commonly referenced alternative.
In non-medical bodybuilding contexts, trestolone is frequently stacked with a DHT-derived compound such as Masteron 100 to help mitigate estrogenic side effects and provide additional hardening effects. A testosterone base such as Cypionate 250 is also commonly referenced, though some users prefer trestolone as a standalone compound due to its potency.
Dosage & Usage
Trestolone 100 mg Dosage & Usage
The information below is provided for educational reference only. Trestolone enanthate is an investigational compound that has never been marketed for medical use; non-medical use falls outside any approved indications and may carry significant health risks.
Typical Dosage Ranges
In non-medical bodybuilding contexts, Trestolone 100 mg is commonly referenced in the range of 100–300 mg per week for intermediate users, with some experienced users referencing up to 400 mg per week. Clinical research studies used substantially lower doses for contraceptive purposes, typically less than 1 mg per day. Because of its long enanthate ester, the weekly total is typically divided into injections administered once or twice per week. The 100 mg/mL concentration means that 1 mL provides 100 mg of trestolone enanthate, allowing for practical injection volumes.
| Use Case | Common Reference Range | Injection Frequency |
|---|---|---|
| Beginner (non-medical) | 100–150 mg / week | Once or twice weekly |
| Intermediate (non-medical) | 200–250 mg / week | Twice weekly |
| Advanced (non-medical) | 300–400 mg / week | Twice weekly |
Stacking & Cycle Considerations
In non-medical bodybuilding contexts, trestolone enanthate is commonly referenced as a standalone compound or stacked with a DHT-derived compound. Dragon Pharma's Masteron 100 is frequently mentioned as a stacking partner to help manage estrogenic side effects. A testosterone base such as Cypionate 250 may also be referenced, though some users prefer to keep testosterone at TRT-level doses when combining with trestolone due to the compound's potency.
Cycle lengths of 6–10 weeks are commonly referenced in non-medical contexts. Because of its long enanthate ester, trestolone clears the body relatively slowly, which means side effects may persist for 2-3 weeks after discontinuation. The compound suppresses endogenous testosterone production rapidly and significantly.
Managing Side Effects
Trestolone is a potent aromatase substrate that converts to 7α-methylestradiol, a highly potent estrogen. This estrogenic activity is the primary side effect concern, with gynecomastia, water retention, and elevated blood pressure commonly referenced in non-medical contexts. Importantly, the methyl estrogen produced by trestolone may bypass standard aromatase inhibitors, meaning that AI drugs like letrozole may not effectively control estrogenic side effects in some users. Some users reference SERMs such as raloxifene for gyno prevention, and prolactin control agents such as cabergoline are sometimes referenced.
Because trestolone does not convert to DHT, hair loss and prostate-related effects are considered less likely compared to testosterone, though individual response varies. Acne is a commonly reported side effect, potentially related to the compound's progestogenic activity and its unique estrogenic profile. Blood pressure and lipid profiles should be monitored during use.
Post-Cycle Therapy (PCT)
After completing a cycle with Trestolone 100 mg, post-cycle therapy is commonly recommended in non-medical contexts to help restore endogenous testosterone production. Because of the long enanthate ester, PCT should begin approximately 2 weeks after the final injection to allow the ester to clear. Agents such as Clomid or Nolvadex are frequently referenced for this purpose. Trestolone is noted for causing significant suppression, so recovery may require extended PCT protocols. Bloodwork and, where possible, medical guidance can help inform recovery strategy.
Important
Individual Response Varies
Dosing strategies, support compounds and recovery protocols should be adjusted based on experience level and bloodwork where possible. The information above is for educational reference and does not constitute medical advice.
Safety & Information
Trestolone Enanthate Safety Information
Trestolone enanthate is an investigational anabolic steroid that has never been marketed for human medical use. It can affect hormonal, cardiovascular, and reproductive function.
Important Safety Information
Trestolone enanthate is an investigational compound that has never been approved or marketed for human medical use. It was studied by the Population Council as a potential male contraceptive, but development was discontinued owing to concerns over side effects, including potential impacts on prostate health and lipid profiles. Non-medical use for bodybuilding or performance enhancement falls outside any approved indication and may carry significant health risks.
Anabolic steroids in general have been associated with serious adverse effects including cardiovascular complications, dyslipidemia, and endocrine disruption. Trestolone's potent estrogenic activity means it carries particular risks related to gynecomastia and fluid retention. Its inclusion on the World Anti-Doping Agency prohibited list underscores its performance-enhancing potential.
Important
Non-Medical Use
Use of trestolone enanthate for bodybuilding or performance enhancement falls outside any approved medical indication. Higher-than-physiologic exposure can increase the risk of serious adverse effects including cardiovascular, hepatic and endocrine complications.
Potential Adverse Effects
Trestolone is a potent aromatase substrate that converts to 7α-methylestradiol, an estrogen with high potency. Estrogenic effects including gynecomastia, water retention, and elevated blood pressure are commonly referenced in non-medical contexts. Importantly, the methyl estrogen produced by trestolone may bypass standard aromatase inhibitors, making management more challenging than with traditional aromatizing compounds. Prolactin elevation may also occur. Acne is a commonly reported side effect, potentially related to progestogenic activity.
Trestolone suppresses gonadotropin release and endogenous testosterone production rapidly and significantly, inducing a state of temporary infertility at sufficient doses. This can lead to sexual dysfunction and testicular atrophy during use. Other potential effects include mood changes, irritability, and lipid profile alterations.
Because trestolone does not convert to DHT due to its 5α-reductase resistance, hair loss and prostate-related effects are considered less likely compared to testosterone. However, individual response varies, and this does not mean the compound is free of androgenic side effects.
Conditions Requiring Medical Evaluation
Trestolone enanthate has not been evaluated for safety in humans with pre-existing medical conditions. Given its potent estrogenic and gonadotropin-suppressing effects, individuals with a history of hormone-sensitive conditions, cardiovascular disease, or hepatic impairment should exercise particular caution. Existing medical conditions should be discussed with a qualified healthcare professional before trestolone is considered.
Monitoring During Use
If trestolone enanthate is used in any context, monitoring of estrogen levels, prolactin, blood pressure, lipid profiles, and hematocrit is important given the compound's known effects. Standard estrogen blood tests may not accurately reflect the methyl estrogen produced by trestolone, making clinical assessment more complex. In non-medical bodybuilding contexts, bloodwork before, during, and after a cycle is commonly referenced as a risk-reduction strategy.
Product Care
Storage & Handling
Keep the vial securely stored and protected from conditions that could compromise the product or container. Store at controlled room temperature and protect from light. Inspect the vial and solution before use and do not use a product that appears damaged, contaminated or otherwise abnormal.
Keep all medications and injectable products out of the reach of children. Follow the storage instructions provided with the product packaging.
Further Safety Information
Shipping & Authenticity
Shipping & Product Authenticity
Trestolone 100 mg by Dragon Pharma is shipped in original manufacturer packaging with discreet, privacy-focused handling.
USA Domestic 3–5 business days
International 10–15 business days
Order Processing 24–48 business hours
Tracking Provided after dispatch
Direct Supply
Discreet Delivery & Original Packaging
The outer shipping package remains discreet, with privacy-focused handling and no unnecessary external product details.
What to Expect
- Orders are processed after payment confirmation
- USA Domestic shipping is typically faster when local stock is selected
- International orders include tracking, though update frequency may vary by destination
- Multiple warehouses may result in separate shipments when applicable
Authenticity Verification
To verify your Trestolone 100 mg product, use the security code on the vial label and cross-check it on the Dragon Pharma official site. Original Dragon Pharma packaging and batch information help reinforce product legitimacy. Given that trestolone is a less commonly produced compound, laboratory verification is particularly valuable for this product.
For complete delivery details, tracking policy, and reshipment terms, please see our Shipping Info page.
Storage
Trestolone 100 mg Storage
Proper storage conditions help preserve formulation stability and overall product integrity throughout shelf life.
Recommended Conditions
Store at controlled room temperature (15–25°C) and protect from excessive heat, moisture, and direct light. Maintaining stable conditions helps preserve the integrity of the oily formulation.
Keep the vial in its original packaging until use. Do not freeze. Before administration, inspect the solution and avoid use if it appears cloudy, discolored, contains particulate matter, or if the vial or seal is compromised.
Keep out of reach of children. Follow proper handling and sterile injection practices when administering the product.
Quick Reference
Do & Don't
- Do store at 15–25°C
- Do keep in original packaging
- Do inspect before each use
- Don't freeze the vial
- Don't expose to direct sunlight
- Don't use if solution looks abnormal
Frequently Asked Questions
Trestolone 100 mg FAQ
Answers to common questions about Trestolone 100 mg, trestolone enanthate, usage considerations, and product strength.
What is Trestolone 100 mg used for?
Trestolone 100 mg contains trestolone enanthate, an investigational compound that was studied as a male contraceptive but never marketed for medical use. In non-medical bodybuilding settings, Trestolone 100 mg is commonly referenced for rapid muscle and strength gains due to its high anabolic potency, though such use falls outside any approved medical indication.
How often should Trestolone 100 mg be injected?
Because of its long enanthate ester and approximately 8-day half-life, trestolone enanthate is typically referenced as being administered once or twice per week in non-medical contexts. The 100 mg/mL concentration means that 1 mL provides 100 mg of trestolone enanthate. Some users prefer more frequent administration for more stable blood levels.
Does Trestolone 100 mg require PCT?
In non-medical bodybuilding contexts, post-cycle therapy is commonly recommended after a trestolone cycle to help restore endogenous testosterone production. Trestolone suppresses gonadotropin release rapidly and significantly. Because of the long enanthate ester, PCT should begin approximately 2 weeks after the final injection. Agents such as Clomid or Nolvadex are commonly referenced for this purpose.
What does trestolone enanthate do?
Trestolone enanthate is a long-acting ester of trestolone that is hydrolyzed in the body to release the active hormone. Trestolone binds to the androgen receptor with high affinity and promotes nitrogen retention and protein synthesis. It does not convert to DHT due to 5α-reductase resistance, but it is a potent aromatase substrate that converts to 7α-methylestradiol, a highly potent estrogen.
How long does Trestolone 100 mg take to work?
Because of its long enanthate ester, trestolone enanthate releases gradually over several weeks. In non-medical contexts, users commonly reference noticing effects after approximately 2 weeks, with full saturation occurring over 4-5 weeks of use. The compound's potency means that effects may become apparent relatively quickly compared to other long-acting AAS.
Is trestolone the best bulking compound?
There is no single compound that is universally best for bulking. Trestolone is commonly referenced in bodybuilding contexts for its exceptional potency and rapid effects. However, its potent estrogenic activity requires careful management, and the methyl estrogen it produces may bypass standard aromatase inhibitors. Other products such as Deca 300 and Cypionate 250 are also referenced for bulking purposes.
What is the difference between Ment 50 and Trestolone 100?
The primary difference is the ester and concentration. Ment 50 contains trestolone acetate at 50 mg/mL, which is a short-acting ester requiring frequent injections. Trestolone 100 mg contains trestolone enanthate at 100 mg/mL, which is a longer-acting ester requiring less frequent injections. Both ultimately provide the same parent hormone, trestolone.
What is the difference between trestolone and testosterone?
Trestolone is significantly more potent than testosterone, with preclinical studies indicating approximately ten times the anabolic potency. Unlike testosterone, trestolone does not convert to DHT and has low affinity for SHBG. However, it converts to a more potent methyl estrogen (7α-methylestradiol) than testosterone does.
Is 100 mg of Trestolone a lot?
A milligram amount cannot be classified as appropriate or excessive without considering the specific context, individual response, and other factors. In non-medical bodybuilding contexts, trestolone enanthate is commonly referenced in the 100–300 mg per week range, divided into one or two injections. Such use falls outside approved indications and requires careful management of estrogenic side effects.
What strength is Trestolone 100 mg?
Trestolone 100 mg is labeled at 100 mg of trestolone enanthate per mL. It is supplied in a 10 mL vial, giving 1,000 mg of total labeled trestolone enanthate content per vial.
Why does trestolone cause more estrogenic side effects?
Trestolone converts to 7α-methylestradiol through aromatization, which is a more potent estrogen than the estradiol produced from testosterone. This means that even at relatively low doses, trestolone can produce significant estrogenic effects such as gynecomastia and water retention. Additionally, the methyl estrogen produced may bypass standard aromatase inhibitors, making management more challenging than with traditional aromatizing compounds.
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Product Information Compound Details
Active Substance Trestolone Acetate Potent 19-nor testosterone derivative (MENT)
50 mg/mLStrength 50 mg/mL
Package 10 mL Vial 500 mg total labeled content
Form Oil-Based Injectable
Carrier MCT Oil
Drug Class Anabolic Androgenic Steroid (19-nor)
Manufacturer Dragon Pharma
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